Table 2.

Strong and moderate CYP3A4 inducers

ClassStrong CYP3A4 inducersModerate CYP3A4 inducers
Antineoplastic Enzalutamide
Apalutamide
Mitotane
Ivosidenib 
Dabrafenib
Lorlatinib
Pexidartinib
Sotorasib 
Other Carbamazepine
Phenytoin
Rifampin 
 
ClassStrong CYP3A4 inducersModerate CYP3A4 inducers
Antineoplastic Enzalutamide
Apalutamide
Mitotane
Ivosidenib 
Dabrafenib
Lorlatinib
Pexidartinib
Sotorasib 
Other Carbamazepine
Phenytoin
Rifampin 
 

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